PREPARATION OF 2-OXA-3-6-DIOXO-9-VINYL-cis-DECALIN SKELETON, A PRECURSOR OF VERNOLEPIN
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چکیده
منابع مشابه
A Simple Method for the Preparation of Cis-(3-Azido-4-Styryl)-2-Azetidinone
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1. The metabolism of cis- and trans-decalin in the rabbit has been investigated. 2. Both hydrocarbons were oxidized to racemic secondary alcohols and excreted as ether glucuronides in amounts equal to about 60% of the dose administered. The principal glucuronides were isolated as triacetyl methyl esters and as sodium salts. 3. cis-Decalin gave rise mainly to (+/-)-cis-cis-2-decalol, together wi...
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In the title compound, C(18)H(20)N(2)O(5), the pyrrolidine ring adopts an envelope conformation with the C atom bonded to the methyl groups as the flap. The dihydro-isoxazole ring is essentially planar (r.m.s. deviation = 0.041 Å) and forms a dihedral angle of 65.19 (6)° with the phenyl ring. In the crystal, neighbouring mol-ecules are linked into chains along [110] by inter-molecular C-H⋯O hyd...
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ژورنال
عنوان ژورنال: Chemistry Letters
سال: 1977
ISSN: 0366-7022,1348-0715
DOI: 10.1246/cl.1977.495